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• Synthesis of Sulfamoyl Ureas from Hexafluoroisopropyl N-Fluorosulfonyl Carbamate
• Nitroxide/Nitric Acid-Promoted Oxidation of Alcohols to Aldehydes and Ketones
• Synthesis of 2-Aminothiophenes Using Piperidinium Borate
• Scalable Synthesis of 4-Bromo-1,2-dimethyl-1H-imidazole
• Primary Benzylic Amines via Copper-Catalyzed Benzylic C(sp3)–H Carbamation
• Novel tert-Butylation of Carboxylic Acids and Alcohols
• Synthesis of Squaric Acid Monoamides as Building Blocks for Drug Discovery
• Synthesis of Glucuronic Acid-Containing Fragments of a Heparin Sulfate Mimetic
• Synthesis of Benzo[b]azepines with a Fluorinated Side Chain
• Mechanochemical Silver-Catalyzed Ring-Opening Fluorination of Cyclobutanols
• Synthesis of Acidiphilamides A–C
• Total Synthesis of Bio-orthogonally Functionalized Securinega Alkaloids
• Visible-Light-Mediated Regioselective Chlorosulfonylation of Acrylamides
• Enantioselective Synthesis of Antispasmodic Drug (R)-Tiagabine
• Synthesis of Trisubstituted Furans from Homopropargylic Alcohols
• Photochemical Flow Synthesis of Pyrazolines from Tetrazoles
• Gold-Catalyzed Stereoselective Synthesis of Polysubstituted Indanes
• Organocatalytic Synthesis of γ-Amino Acid Precursors
• Oxidation of α-CF3 and Other Secondary Alcohols to Ketones Using a Nitroxide Catalyst
• Regioselective Synthesis of 5-Substituted Pyrazoles
• Synthesis of the Proposed Structure of Cryptoconcatone H
• One-Step and Gram-Scale Synthesis of Caffeine-d9
• Bromothiolation of Internal Alkynes
• Photooxidation of Toluene Derivatives into Carboxylic Acids
• One-Pot Synthesis of Diaryl Sulfonamides via Metal Catalysis
• Gram-Scale Synthesis of Substituted Triarylmethanes
• Synthesis of [10]Cycloparaphenylenes and their Binding to C60
• Improved Scalable Synthesis of the (S,S)-DACH-Ph Trost Ligand
• Rh(II)-Catalyzed N–H Amination of Aliphatic Amines and α-Amino Acids
• Novel Nickel-Catalyzed Synthesis of (Trifluoromethyl)quinolines
• Synthesis of Quaternary α-Fluoronitriles from Monofluorolkenes
• Stereoselective Synthesis of (–)-Heliannuol E
• General Entry to Pyrazolo[3,4-b]pyridine-3-carboxamides
• Seven-Step Synthesis of (±)-epi-Costunolide
• Total Synthesis of a Microbiologically Important Pentasaccharide
• Synthesis of the Selective Serotonin 2A Receptor Agonist 25CN-NBOH
• Synthesis of Ar-SF4Cl and Ar-SF5 Compounds from Arylphosphorothiolates
• Entry to N-Protected Serine/Threonine-Derived Weinreb Amides
• Oxa-(4+4)-Cycloaddition Entry to Oxazocine Scaffolds
• Concise Total Synthesis of (+)-Aphanorphine
• Synthesis of Allyl Aryl Sulfones from Morita–Baylis–Hillman Adducts and Thiosulfonates
• Fe(III)-Catalyzed Synthesis of 1-Chalcogenylated Naphthalene Derivatives
• Catalytic Synthesis of Olivetol and Derivatives
• Nickel-Catalyzed Synthesis of Benzofuran Derivatives
• Synthesis of Fluorenone-Fused Coumarins
• Stereoselective Synthesis of the Cotylenin A Aglycone Carbon Skeleton
• Novel Entry to Fluorinated Cyclopropanes
• Ni-H-Catalyzed Isomerization-Induced Cleavage of Allyl Ethers
• Continuous Photochemical Benzyne-Forming Process
• Copper-Catalyzed Ring Expansion of Vinyl Aziridines
• Synthesis of Constrained Benzoxazepines and Imidazopyrazines
• Synthesis of N-Aryl-1,2,3,4-tetrahydroisoquinolines
• A Molecular Stereostructure Descriptor for Asymmetric Catalysis
• A Catalytic One-Pot Synthesis of Indolyl Cyclobutanones
• Vitamin B12-Photo-Catalyzed Dicarbofunctionalization of Bromoalkenes
• Scalable Synthesis of Thiazole Peptide Macrocycles
• Synthesis of Optically Active Maresin 2
• Decarbonylative Alkynylation of Acyl Fluorides
• First Total Synthesis of the Alkaloid Clausenalansine A
• Synthesis of 4,5-Diaryl-2H-1,2,3-triazoles
• Diastereoselective Total Synthesis of (±)-Parvistemonine A
• Synthesis of Thienyl Thioethers and Thieno[3,2-b]thiophenes
• Synthesis of an Azabicyclo[3.1.0]hexanone Drug Candidate
• Redox-Neutral C1-Alkynylation of Tetrahydroisoquinolines
• Synthesis of Secondary Alcohols from Alkynes in Water
• Synthesis of Fused-ring Heptacyclic Pyrrolidines
• Peptide Synthesis with α,α-Difluoro-β-Lactams
• Synthesis of 13,19,20-Trihydroxy Docosahexaenoic Acid Stereoisomers
• Propargylation of Diaryl Azo Compounds
• Total Synthesis of Phyllanemblinin B
• Synthesis and Structure of 1-Substituted Semithioglycolurils
• Copper-Catalyzed Stereoselective Synthesis of 2-Deoxygalactosides
• Synthesis of Alkyl-methyl/ethyl Derivatives from N-(Acyloxyalkyl)phthalimides
• Synthesis of N-Substituted Ureas from Primary Amides
• Regioselective Synthesis of 3,5-Disubstituted Pyrazoles
• Synthesis of Hybrid Chromone/Coumarin 3-Halo-1H-indenes
• Annulation Approach to Tetrahydro-1,2,4-triazinecarboxylate Esters
• Scalable Synthesis of Sphingomyelins
• Synthesis of Polycyclic Indolines
• Diels–Alder Based Approach to Prenyleudesmane Diterpenoids
• Total Synthesis of Glycosyl Flavonoids
• Total Synthesis of Asparenydiol
• Synthesis of the Enantiomers of Thioridazine
• Novel Synthesis of Benzoxazoles and Benzimidazoles
• A Study of Samarium(II)–Water Allylic Benzoate Reductions
• Formal Synthesis of Pseudolaric Acid B
• Metal-Free Synthesis of Hindered 3-Azoindoles
• Multigram Deoxofluorination of β-Keto Esters with Sulfur Tetrafluoride
• A Radical-Chemistry Approach to 2-Arylquinolines
• Novel 2-Substituted Analogues of (–)-Pentenomycin I
• Detailed Comparison of Ni vs. Pd in Cross-Coupling Catalysis
• Synthesis of Sulfonylisoureas via Sulfo-Click Reactions
• Selenium Tetrachloride Catalyzed Iodination of (Hetero)Arenes
• Pd-Catalyzed Synthesis of N-Allyloxypyrrolidinediones
• A Novel Approach to Diarylated Esters and Phosphonates
• One-Pot Access to 2-Aryl-3-(arylmethyl)chromones
• Benzoazepinoindoles – A New Class of Heterocycles
• Metal-Free Hydroamination of Alkynes
• 1,2,4,5-Tetrazine Derivatives from Arylsulfonylhydrazones
• Mono- and Dihalogenation of 2-Aminopyrazine
• Novel Approach to Antihistamine-type Scaffolds
• Poster Prize awarded at ISySyCat 2019
• An Improved Synthesis of 2,5-Disubstituted Tetrazoles
• Total Synthesis of Shensongine A
• Synthesis of Novel Imidazothiadiazoles
• Cu(II)-Catalyzed Beckmann Rearrangement of Ketones
• Allylic C–H Alkynylation via Copper Photocatalysis
• Synthesis of Dumbbell-like Amine-Functionalized Bis-C60 Fullerene
• It was not tricyanomethane, after all…
• Total Syntheses of (+)-Alexine and Related Alkaloids
• Poster Prize awarded at Bioheterocycles 2019
• Photoredox Fischer Indole Synthesis
• Synthesis of Resolvins and Derivatives
• Poster Prize awarded at Twente / Mainz Symposium
• First Total Synthesis of Artekeiskeanol A, C and Altissimacoumarin D
• Iodoglycosylation and Iodocarboxylation of Glycals
• Gold(III)-Catalyzed Synthesis of N,N-Aryl,Benzyl-amines in Water
• Synthesis of Fatty Acid Intermediates via Hudrlik–Peterson Reaction
• Recyclable Graphene Oxide Nanosheet Supported Catalyst
• A Stereoselective Synthesis of the ACE Inhibitor Trandolapril
• New Entry to 3-Arylglutaconic Acid Derivatives
• Electrochemical C(sp³)–H Fluorination
• Asymmetrische Synthese von α-Hydrazinoketonen
• Synthese von (–)-Boschnialacton und γ-Lycoran
• Synthesis of the ABC-Ring System of Various Alkaloids
• Regioselective Halogenation of Coumarins
• Synthesis of 4-(Arylmethyl)proline Derivatives
• Efficient Synthesis of a 5α-Reductase Inhibitor
• Epoxidation of a Cyclic Allyl-Amine by a Bifunctional Peracid
• Radiochemical Synthesis of 2-[18F]Fluorophenylalanine
• Asymmetric Mannich-Type Reaction of an α-Trifluoromethyl Amide
• Chemoselective Aerobic Oxidation of Benzylic Alcohols
• One-Pot Reductive Conversion of Aldehydes into Acetic Esters
• Visible-Light-Induced Adamantylation of Azoles
• Synthesis of Protected Stereodefined 5-Aminomethylprolines
• Synthesis of Thiophene-Fused 1,10-Phenanthrolines
• Synthesis of 8-Oxabicyclo[3.2.1]octanes
• Asymmetric Synthesis of Netarsudil
• Borylated Cyclohexenes via Suzuki–Miyaura/Diels–Alder Cascade
• Synthesis of 1-Alkylisoquinolines via Radical Cyclization
• Biphenyls via Cross-Coupling of Arenediazonium Salts
• Synthesis of Anthraquinones via Pd-Catalyzed Acylation
• Synthesis and Applications of 4-Chloro-2-(trichloromethyl)pyrimidines
• Catalyzed Conversion of Aldehydes into Nitriles
• Synthesis of Aryl/Heteroaryl Amides via Nitriles Hydration
• Stereospecific Amination of Alkylboronic Esters
• Metathesis Reactions for Accessing β-Amino Acid Derivatives
• Selective Preparation of C2v-Symmetric Hexaphenylbenzenes
• Stereoselective Oxidation of Titanium(IV) Enolates with Oxygen
• Ring-Closing Metathesis Entry to Dienamide Heterocycles
• New Dipeptide Organocatalysts for Aldol Reactions
• A Biomimetic Synthesis of des-Hydroxy Paecilospirone
• Monitoring Solid-Phase Reactions with Thin-Layer Chromatography
• Multi-Component Synthesis of N-Unsubstituted 1,2,3-Triazoles
• Organocatalytic Enantioselective Synthesis of 1,3-Disubstituted Allenols
• Improved Synthesis of Guanine Quadruplex Ligand Phen-DC3
• C–H Alkylation of Heteroarenes with Alkyl Bromides
• Synthesis of Nepetoidin B
• Synthesis of 2-Azabicyclo[n.2.0]alkane-Derived Building Blocks
• Novel Approach to Organo-Phosphinates and Phosphonates
• Conceptually New Approach to Ellipticine and the Oxoaporphine Core
• Difluoro(phenylsulfanyl)methane as a Formylating Agent
• Synthesis of a Gallium Complexing Agent used in PET Tracers
• Increasing Tetrazine Reactivity in the IEDDA Reaction
• Multicomponent Entry to Polysubstituted 2-Aminopyrroles
• Palladium-Catalyzed Synthesis of Arylgermanium Compounds
• Synthesis of 1-Monosubstituted 1,2,3-Triazoles
• Continuous-Flow Synthesis of Chiral 1,2-Diamino Derivatives
• New Synthesis of Azulene
• A Synthesis of S,S-DICHED Catalyst for Matteson Homologations
• Novel Oxazole-Containing Amino Acids
• B-Ring Contraction in Steroids via Benzilic Acid Rearrangement
• Photoredox Synthesis of Arylhydroxylamines
• Unsymmetrical Biheteroaryls via Suzuki–Miyaura Cross-Couplings Using an Air-Stable Pre-Catalyst
• Unsymmetrical Biheteroaryls via Suzuki–Miyaura Cross-Couplings Using an Air-Stable Pre-Catalyst
• Mechanistic Insight on the Bromocycloetherification of Alkenes
• Synthesis of Arylalkynes from Diaryl Sulfoxides
• SYNLETT Editorial Board Welcomes New Members
• New Heptitol Derivatives as Potential Antibacterials
• New Entry to Cyclopentyl Aryl Ketones via Photoredox Catalysis
• Iodide-Catalyzed Carbonylation–Benzylation of Benzyl Chlorides
• Synthesis of Functionalized Rubicenes
• Pd-Catalyzed Synthesis of ortho-Fluorodiarylmethanes
• Novel Entry to Tetraarylmethanes
• Synthesis of N-Arylsulfonamides
• Monofluoro Aryl Acetates via Copper Catalysis
• Enaminones via Palladium-Catalyzed Four-Component Carbonylation
• Trifluoromethylation of Highly Functionalized Heteroarenes: Flow to the Rescue
• Novel Synthesis of Aryl Cyclopropylketones
• Total Synthesis of Lagerstannin C
• New Synthetic Access to Ethers
• Stereoselective Cyclopropanation of (–)-Levoglucosenone Derivatives
• Microwave-Promoted Synthesis of 4-Arylpyrimidines in Water
• Protein Synthesis and Crystallization of Bowman–Birk Protease Inhibitors
• Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins
• Synthesis of 3,5,7-Trisubstituted Indoles
• Rhodium(III)-Catalyzed Sulfonamidation of Azoxybenzenes
• Synthesis and Properties of 2-Oxa-6-azaspiro[3.3]heptane Sulfonate Salts
• Metal-Free Primary Amination of Potassium Aryltrifluoroborates and Phenylboronic Acids
• Synthesis of a Ubiquitinated Histone Mimic Bearing a New Thioether Linkage
• Organocatalytic Synthesis of non-Racemic Oxazolines from Isocyanoacetate and α-Keto Esters
• Catalytic Asymmetric α-Hydroxylation of 3-Substituted Oxindoles with Hydrogen Peroxide
• Synthesis of Benzo[e]azolo[1,3]oxazines
• Preparation of 3-Aminoimidazo[1,2-a]pyrazines
• [3+2] Cycloaddition of Azomethine Ylides
• Synthesis of N,O-Nucleosides via Ene Reaction
• Bunte Salts as Thiolating Reagents for Alkenes
• Synthesis of Fused Naphthobenzofurans
• New Entry to Tetrahydropyrazolopyrazolones via [3+2] Cycloaddition
• Enantiocontrolled Synthesis of Non-racemic γ-Acetoxyallylboronates
• Asymmetric Aldol Reactions with a Dual Catalyst System
• Multistep Continuous-Flow Synthesis of (–)-Oseltamivir
• Synthesis of the Siderophore Erythrochelin
• New Parallel Synthesis of Di(hetero)arylamides
• Augmented Reality as an Enabling Tool in Organic Chemistry
• Lanthanum-Catalyzed Olefination of Benzylamines with 2-Methylquinoline via Tandem Oxidation/Benzylidene Addition
• Efficient Access to the Structural Core of Annonaceous Acetogenins
• Synthesis of α-Arylglycines and Other α-Amino Acid Derivatives
• New Synthesis of Morpholines and Benzoxazines
• Synthesis and Structural Revision of a γ-Lactone Polyketide of Fungal Origin
• 2-Alkynyl-1,4-cyclohexadienes via a Diels–Alder Reaction
• Aryltrimethylgermanes for the Arylation of Amines and Amides
• Samarium(II)-Promoted Synthesis of 2-Azabicycles
• First Total Synthesis of Dermocanarin 2
• Synthesis of Enantiopure tert-Butylmethylphosphine–Boranes
• Total Synthesis of δ-Sanshool and Analogues
• Novel Entry to Peptides Incorporating Tryptophan and Analogues
• Photoredox Catalysis for a Novel Access to Pentafluorosulfanyl Compounds
• Novel Substrates for Desymmetrization Processes
• Enantiopure Monomethylated L-Arginine and L-Ornithine
• Iodo- and Chloroamination of Enecarbamates
• Enantioselective N-Functionalization of Pyrroles
• Novel Fluorescently Labeled Amino Acids
• Synthesis of Enantiomerically Pure β-Methoxytyrosine
• Novel Route to Aromatic Hydrazines via Cu-Catalyzed Addition of Arylboronic Esters to Azodicarboxylates
• Novel Synthesis of Orthogonally Protected Diazaspiro[3.4]octane Analogues
• Trityl Group Deprotection from Tetrazoles
• Synthesis of Cyclotribenzoin
• Synthesis of New Chiral Diaryliodonium Salts
• Synthesis and Analysis of Macrocyclic Peptides with 3₁₀-Helical Structure
• Total Synthesis of (+)-Clavulatriene A
• Biologically Important Phosphotriesters by Organocatalysis
• New Potential Organic Semiconductors

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